Аннотация:Data on methods of the synthesis of conformationally restricted analogs of γ-aminobutyric acid (GABA) are systematized in the review. Approaches to the synthesis of different types of conformationally restricted GABA analogs are presented: γ-aminobutenoic acids, aminocycloalkanecarboxylic acids, carboxy-substituted azetidines, prolines, amino acids containing aromatic (heterocyclic including) fragments.